About and Introduction

• Abstract - Open Access

  Prefacio

  Santos, Alcindo A. Dos

  PDF - p-326-327

• Abstract - Open Access

  About the Royal Society of Chemistry

  Magalhaes, Elizabeth; Jones, Ray

  PDF - p-309-309

• Abstract - Open Access

  Design and applications of selective reactions of olefins

  Grubbs, Robert H.

  PDF - p-310-310

Keynote

• Abstract - Open Access

  Selectivity in Metal-Catalyzed C–H Functionalizations

  Ackermann, Lutz

  PDF - p-316-316

• Abstract - Open Access

  Assembly Line Synthesis

  Aggarwal, Varinder

  PDF - p-317-317

• Abstract - Open Access

  NEW HORIZONS OF GOLD CATALYSIS

  Hashmi, A. Stephen K.

  PDF - p-318-318

• Abstract - Open Access

  Preparation of chiral prim-, and sec-amines employing biocatalysts

  Kroutil, Wolfgang; Simon, Robert C.; Busto, Eduardo; Richter, Nina; Tauber, Katharina; Fuchs, Christine S.; Pressnitz, Desiree; Fischereder, Eva-Maria; Lechner, Horst; Zepeck, Ferdinand

  PDF - p-319-319

• Abstract - Open Access

  Target Synthesis Directed Methodology Development

  Ma, Dawei

  PDF - p-320-320

• Abstract - Open Access

  Strategies and Tactics for Synthesis Inspired by Complex Alkaloids

  Sarpong, Richmond

  PDF - p-321-321

• Abstract - Open Access

  Catalytic oxidations by metal nanoparticles: Pd, Au and AuPd core-shell nanoparticle catalysts

  Rossi, Liane M.; Silva, Tiago A. G.; Teixeira-Neto, Erico; Lopez, Núria

  PDF - p-322-322

• Abstract - Open Access

  Late-Stage Fluorination

  Ritter, Tobias

  PDF - p-323-323

• Abstract - Open Access

  Synthesis and Functions of Biomimetic Helical Polymers and Oligomers

  Yashima, Eiji

  PDF - p-324-324

• Abstract - Open Access

  Borylation, Silylation, Fluorination and Fluoroalkylation

  Hartwig, John F.

  PDF - p-325-325

• Abstract - Open Access

  Continuous Chemical Synthesis in Flow

  Baxendale, Ian R.

  PDF - p-326-326

• Abstract - Open Access

  The Baylis-Hillman reaction: Our vision and experience

  Basavaiah, D.

  PDF - p-327-327

• Abstract - Open Access

  Mechanistic Studies on the Copolymerization of Epoxide with Carbon Dioxide

  Nozaki, Kyoko

  PDF - p-328-328

• Abstract - Open Access

  Enantioselective Heck Reactions with Aryldiazonium Salts. Challenges and Synthetic Opportunities

  Correia, Carlos Roque Duarte

  PDF - p-329-329

Young Talents

• Abstract - Open Access

  Catalysis and mechanistic investigation with ionically-tagged reagents

  Neto, B. A. D.

  PDF - p-311-311

• Abstract - Open Access

  Chemoselective Transformations for Bioimaging and Targeted Therapeutics

  Bernardes, Gonçalo J. L.

  PDF - p-312-312

• Abstract - Open Access

  COMPUTATIONALLY INEXPENSIVE GIAO 13C NMR CALCULATIONS COUPLED WITH ARTIFICIAL NEURAL NETWORK PATTERN RECOGNITION AS A NEW STRATEGY TO AVOID CHASING MOLECULES THAT WERE NEVER THERE

  Sarotti, Ariel M.

  PDF - p-313-313

• Abstract - Open Access

  Directing Group Enhanced Carbonylative Ring Expansions of Amino Substituted Cyclopropanes

  Bower, John F.

  PDF - p-314-314

• Abstract - Open Access

  α,β-Unsaturated Diazoketones as Useful Platforms in the Synthesis of Pyrrolidine, Piperidine and Indolizidine Alkaloids

  Burtoloso, Antonio C. B.

  PDF - p-315-315

Abstracts

• Abstract - Open Access

  An efficient and reusable palladium nanocatalyst in C-C bond forming cross-coupling reactions

  Ganapathy, D.; Sekar, G.

  PDF - p-1-1

• Abstract - Open Access

  Synthesis of non-peripherally substituted phthalocyanines with alkylsulfanyl groups

  A., Cidlina; V., Novakova; P., Zimcik

  PDF - p-2-2

• Abstract - Open Access

  Electrochemical dimerization of benzyl chloride on a powder cathode of silver, graphite or silver-graphite mixture

  Souza, Ronny F. M.; Areias, Madalena C. C.; Navarro, Marcelo; Laurent, Michel; Léonel, Eric; Cachet-Vivier, Christine; Bieber, Lothar W.

  PDF - p-3-3

• Abstract - Open Access

  Studies toward the first total synthesis of Floribundane B

  Silva, João V. S.; Resck, Inês; Machado, Angelo H. de L.

  PDF - p-4-4

• Abstract - Open Access

  Organic acids as efficient catalysts for microwave-assisted synthesis of xanthenones

  Terra, Bruna Silva; Fátima, Ângelo de

  PDF - p-5-5

• Abstract - Open Access

  A New Method of Spiroketalization via Cascade Oxidative Dearomatization

  Shirley, Harry J.; Bray, Christopher D.

  PDF - p-6-6

• Abstract - Open Access

  Highly Selective Tandem Nitrone Formation/1,3-Dipolar Cycloaddition Catalyzed by Ruthenium Porphyrin

  Reddy, Annapureddy Rajasekar; Guo, Zhen; Siu, Fung-Ming; Lok, Chun-Nam; Liu, Fuli; Yeung, Kai-Chung; Zhou*, Cong-Ying; Che, Chi-Ming

  PDF - p-7-7

• Abstract - Open Access

  Development of Methodology for Glycopeptide Enrichment

  Caixeta; Vanessa; Westerlind; Ulrika

  PDF - p-8-8

• Abstract - Open Access

  Regioselective synthesis of 1,3- and 1,5-substituted pyrazoles and pyrazolynes analogous of Celecoxib

  Zanatta, Nilo; Lobo, Marcio M.; Canova, Bruna; Bonacorso, Helio G.; Martins, Marcos A. P.

  PDF - p-9-9

• Abstract - Open Access

  3H-1,2-dithiole-3-thione to (E)-3-[1-(alkylthio)alkylidene]-3H-1,2- dithiole transformation: theoretical and experimental studies

  Couto, Marcos; Cabrera, Mauricio; Echeverría, Gustavo A.; Piro, Oscar E.; González, Mercedes; Cerecetto., Hugo

  PDF - p-10-10

• Abstract - Open Access

  Synthesis, Properties, and Application of Novel Spirocondensed Dithienogermoles

  Wu, L.; Reichert, T.; Saragi, T.P.I.; Fuhrmann-Lieker, T.; Salbeck, J.

  PDF - p-11-11

• Abstract - Open Access

  Synthesis of Dipyrone Metabolites and Evaluation of their Antipyretic Effect

  Vaz, Artur; Aguiar, Fernando A.; Malvar, David C.; Souza, Gloria E. P.; Clososki, Giuliano C.

  PDF - p-12-12

• Abstract - Open Access

  Directed Magnesiation of Haloaromatics Oxazolines using the Tetramethylpiperidylmagnesium Reagents TMPMgCl.LiCl

  Batista; J.H.C.; Santos; F.M.; Silva; S.C.; Oliveira; A.R.M.; Clososki; G.C

  PDF - p-13-13

• Abstract - Open Access

  Efficient synthesis via molecular sieve of 3-(pyrimidin-2yl)- thiazolidinones

  Ribeiro; C.S.; Jr, Campos; J.C.; Bierhals; M.P.; Freitag; R.A.; Cunico; W.; Siqueira; G.M.

  PDF - p-14-14

• Abstract - Open Access

  Biginelli reaction using lemon juice as catalyst under microwave irradiation

  *, Thalita Corrêa C. de Oliveira; Souza, Andrea Luzia F. de

  PDF - p-15-15

• Abstract - Open Access

  Chiral Brønsted Acid Catalyzed Highly Stereoselective Mannich-type reaction of Azlactone with Aldimines

  Gonçalves, Vanessa P.; Justo, Rodrigo M. S.; Amarante, Giovanni W.

  PDF - p-16-16

• Abstract - Open Access

  New Synthesis for norbornene from 4-amoniantipyrine

  Silveira, Ingridhy Ostaciana Maia Freitas da; Winck, Cristiane Regina; Oliveira, Paola Dias de; Gomes, Roberto da Silva; Lima, Denis Pires de; Beatriz, Adilson

  PDF - p-17-17

• Abstract - Open Access

  Methodological study of the classic Claisen rearrangement in Morita-Baylis-Hillman adducts

  Rodrigues, Tiago C. A. F.; Machado, Wender Alves da Silva* e Angelo H. L.

  PDF - p-18-18

• Abstract - Open Access

  Synthesis of Isoxazolic analogues derivatives of Grandisin and Veraguensin neolignans with anti-leishmania and antitrypanosomal activities

  Soares, Ozildéia; Hurtado, Gabriela R.; Viana, Luiz H.; Albuquerque, Sérgio de; Baroni., Adriano C. M.

  PDF - p-19-19

• Abstract - Open Access

  An experimental and theoretical study of the cycloaddition reactions of carbomethoxy-para-benzoquinones with 6,6-dimethyl-fulvene

  Servilha, Bruno M.; Donatoni, Maria C.; Oliveira, Kleber T. de; Ferreira, Marco A. B.; Brocksom, Timothy J.

  PDF - p-20-20

• Abstract - Open Access

  Synthesis and antioxidant activity of nitroaryl-1,2,3-triazoles

  Valença, Wagner O.; Costa, Pollyanna L. F. da; Freitas, Jucleiton J. R. de; Silva, Tânia Maria S. da; Oliveira, Ronaldo N. de

  PDF - p-21-21

• Abstract - Open Access

  Synthesis and evaluation against Trypanosoma cruzi of naphthoquinone-containing triazoles

  Diogo, Emilay B. T.; Dias, a Gleiston G.; Valença, Wagner O.; Camara, Celso A.; Silva, Mauro G. da; Oliveira, Ronaldo N. de; Menna-Barreto, Rubem F. S.; Castro, Solange L. de; Júnior, Eufrânio N. da Silva

  PDF - p-22-22

• Abstract - Open Access

  Cycloadducts Synthesis and Relative Stereochemistry Determined by NMR and DFT-GIAO calculations

  Resende*, Gabriela da C.; Alvarenga, Elson S. de

  PDF - p-23-23

• Abstract - Open Access

  Exploring the enantioselective Heck-Matsuda reaction with electron-rich endocyclic olefins – 2,3-dihydrofuran asymmetric arylation

  Schwalm, Cristiane Storck; Correia, Carlos Roque Duarte

  PDF - p-24-24

• Abstract - Open Access

  Synthesis and Evaluation against Mycobacterium tuberculosis of Phenazine-triazole-linked from ortho-Naphthoquinones

  Jardim, Guilherme A. M.; Dias, Gleiston G.; Diogo, Emilay B. T.; Silva, Diego A. C.; Rodrigues, Bernardo L.; Cantos, Jéssica; Silva, Pedro E. A.; Júnior, Eufrânio N. da Silva

  PDF - p-25-25

• Abstract - Open Access

  An expeditious approach to tetrahydroindolizines from Morita- Baylis-Hillman Adducts

  Teodoro, Bruno V. M.; Correia, José Tiago M.; Coelho, Fernando

  PDF - p-26-26

• Abstract - Open Access

  A simple access to ionic liquids using N-substituted imidazole derivatives from Morita-Baylis-Hillman adducts

  Santos, Marilia S.; Jr., Manoel T. Rodrigues; Coelho, Fernando

  PDF - p-27-27

• Abstract - Open Access

  Benzothiadiazole-triazole-linked biologically active lapachone derivatives: Antitumoral activity and bioimaging application

  Cruz, Eduardo H. G. da; Carvalho, Pedro H. P. R.; Silva, Diego A. C. da; Diogo, Emilay B. T.; Pessoa, Claudia; Coêlho, Bruno; Neto, Brenno A. D.; Júnior, Eufrânio N. da Silva

  PDF - p-28-28

• Abstract - Open Access

  Synthesis and spectroscopic characterization of urea/thiourea derivatives for potential optical sensors application

  Silva*, Claudia Brito da; Rodembusch, Fabiano Severo

  PDF - p-29-29

• Abstract - Open Access

  Synthesis of 2,3-Diaryl-2-azabicyclooctanones derivatives by multicomponent reaction promoted by Nb(OEt)5.

  Silva, Bruno Henrique Sacoman Torquato da; Martins, Lucas Michelão; Silva-Filho., Luiz Carlos da

  PDF - p-30-30

• Abstract - Open Access

  Phenanthrenequinone chlorination with trichloroisocyanuric acid

  Azeredo, Sirlene Oliveira Francisco de; Figueroa-Villar, José Daniel

  PDF - p-31-31

• Abstract - Open Access

  Selective semi-hydrogenation of propargylamines using palladium magnetic nanocatalyst

  Uberman, Paula M.; Costa, Natalia J. S.; Albuquerque, Joao L. P.; Santos, Alcindo A. Dos; Rossi, Liane M.

  PDF - p-32-32

• Abstract - Open Access

  Selective oxidative aromatization of polyfunctionalized trifluoromethyl substituted chromenones by microwave irradiation

  Cavinatto, Susiane; Navarini, Jussara; Wiethan, Carson W.; Junges, Andrizia F.; Pittaluga, Everton P.; Luz, Fábio M.; Paim, Gisele R.; Martins, Marcos A. P.; Zanatta, Nilo; Bonacorso., Helio G.

  PDF - p-33-33

• Abstract - Open Access

  Formal γ-alkynylation of ketones via Pd-catalyzed C-C cleavage

  Ziadi, Asraa; Correa, Arkaitz; Martin, Rubén

  PDF - p-34-34

• Abstract - Open Access

  Metal-catalyzed direct carboxylation of unactivated alkyl halides with CO2

  Liu, Yu; Martin, Ruben

  PDF - p-35-35

• Abstract - Open Access

  General pathways for obtainment of halo-containing 1,8- naphthyridines,1,8-naphthyridin-2(1H)-ones and their derivatives

  Andrighetto, Rosália; Bonacorso, Helio G.; Stefanello, Felipe S.; Martins, Marcos A. P.; Zanatta, Nilo

  PDF - p-36-36

• Abstract - Open Access

  New strategy for the synthesis of Bromacil and their analogous

  Zanatta, Nilo; Santos, Josiane M. dos; Silveira, Alessandra da; Bonacorso, Hélio G.; Martins., Marcos A. P.

  PDF - p-37-37

• Abstract - Open Access

  Synthesis of (–)-(R)-angustureine by formal alkynylation of a chiral ß-amino ester

  Muñoz*, Gaspar Diaz; Dudley, Gregory B.

  PDF - p-38-38

• Abstract - Open Access

  Synthesis of naphthoxazole derivates from lapachol and their isolation by countercurrent chromatography

  Rio, Karina P. DeI; Leitão, Gilda G.; Moura., Kelly C. Gallan de

  PDF - p-39-39

• Abstract - Open Access

  Enzymatic kinetic resolution of methyl 2-methyl-4-oxopentanoate

  Ferreira, Edgard A.; Omori, Álvaro T.; Cunha, Rodrigo L. O. R.

  PDF - p-40-40

• Abstract - Open Access

  Synthesis of C7−C31 fragment of (−)-cryptocaryol A

  Kuroishi, Paula K.; Jr., Emílio C. de Lucca; Dias, and Luiz C.

  PDF - p-41-41

• Abstract - Open Access

  Studies on the use of Poliethyleneglicol (PEG) in Heck Oxyarylation Reaction for the Synthesis of Deoxy Pterocarpans and Analogs

  Moraes, Paula de F. de; Gaspar, Francisco V.; Leão, Raquel A. C.; Costa, Paulo R. R.

  PDF - p-42-42

• Abstract - Open Access

  Synthesis of new hemilabile ligands based on phosphinic amide and pyrazolo[1,5-c]quanazoline moieties Applications in coordination chemistry

  Marra, Roberta K. F.; Bernardino, Alice M. R.; Souza, Marcos C. de; Romeiro, Gilberto A.; Iglesias, María J.; López-Ortiz, Fernando

  PDF - p-43-43

• Abstract - Open Access

  Photochemical activity of a key donor-acceptor complex can drive stereoselective catalytic a-alkylation of aldehydes

  Arceo, E.; Jurberg, I. D.; Álvarez-Fernández, A.; Melchiorre, P.

  PDF - p-44-44

• Abstract - Open Access

  Design of Experiments Applied to Heck-Matsuda Arylations. Optimizing the Synthesis of Resveratrol, DMU and Stilbene Derivatives

  Correia, Carlos Roque Duarte; Perez, Carla Cristina

  PDF - p-45-45

• Abstract - Open Access

  CHELATOR-PEPTIDE CONJUGATE AS PROTECTOR AGAINST IRON-INDUCED TOXICITY

  Goswami, D.; Vitorino1, H. A.; Machini, M. T.; Esposito, B. P.

  PDF - p-46-46

• Abstract - Open Access

  Studies toward an indanone-based hybrid with potencial AchE inhibition to treat Alzheimer’s disease

  Chierrito, Talita Perez Cantuaria; Carvalho, Marcelo Rodrigues de; Carvalho., Ivone

  PDF - p-47-47

• Abstract - Open Access

  New modular structures constructed by click chemistry

  Valdomir, Guillermo; Padrón, José M.; Padrón, Juan I.; Martín, Víctor S.; Davyt, Danilo

  PDF - p-48-48

• Abstract - Open Access

  Unexpected dimerization of a nitrobenzyl chloride under basic conditions

  Santos, Giovanna C.; Macedo, Jéssica B.; Lopes, Marcela S.; Pádua, Rodrigo M. de; Oliveira, Renata B.

  PDF - p-49-49

• Abstract - Open Access

  Asymmetric Arylation of Indenes via Heck-Matsuda Reaction

  Carmona, Rafaela C.; Correia, Carlos Roque D.

  PDF - p-50-50

• Abstract - Open Access

  Preparation of New Prenylated (E)-Chalcones

  Santos, *Mariana Bastos dos; Gullo, Fernanda Patricia; Dutra, Luiz Antonio; Mendes-Giannini, Maria José Soares; Fusco-Almeida, Ana Marisa; Regasini, Luis Octávio

  PDF - p-51-51

• Abstract - Open Access

  Synthesis and citotoxicity activity of new aza-analogues of angucyclinones from (-)-shikimic acid

  Cuellar, M; Quiñones, N; Villena, J; Salas, C.

  PDF - p-52-52

• Abstract - Open Access

  Synthesis of the C1-C13 fragment of Nhatrangin A

  Polo, Ellen Christine; Dias, Luiz Carlos

  PDF - p-53-53

• Abstract - Open Access

  Synthesis of fluorinated aminosugars Positron Emission Tomography diagnostic studies

  Nunes, Paulo Sérgio Gonçalves; Bernades, Emerson Soares; Carvalho, Ivone

  PDF - p-54-54

• Abstract - Open Access

  Investigation of proline derivatives for the efficient organocatalysis of an Aldol type reaction in supercritical CO2

  Cassaro, R. F.; Sakae, G.; Takata, L.M.; Santos, A. dos; Gariani, R. A.; Bazito, R. C.

  PDF - p-55-55

• Abstract - Open Access

  Iodination of Benzylanilines with Potassium Dichloroiodate

  Mota, George J. M.; Garden, Simon J.

  PDF - p-56-56

• Abstract - Open Access

  Synthesis of the C10−C22 Fragment of Marinisporolide A

  Júnior, Emílio Carlos de Lucca; Dias, Luiz Carlos

  PDF - p-57-57

• Abstract - Open Access

  Studies in Organocatalyzed Direct Aldol Reactions under Solvent-Free Conditions

  Silva, Rúbia Yano da; Aguilar, Andréa Maria

  PDF - p-58-58

• Abstract - Open Access

  Simple and efficient synthesis of triazole-based iminosugars with potential anti-glucosidase activity

  Aragão-Leoneti, Valquiria; Carvalho, Ivone

  PDF - p-59-59

• Abstract - Open Access

  Synthesis of Six-membered Ring Analogues of RK-682 and Meldrum’s acid derivatives. Evaluation on the Inhibition of Protein Tyrosine Phosphatases

  Carneiro, Vânia M. T.; Trivella, Daniela B. B.; Aparicio, Ricardo; Pilli, Ronaldo A.

  PDF - p-60-60

• Abstract - Open Access

  Enantioselective catalysis from Pseudomonas cepacia on the kinetic resolution by different reactors

  Manoel*, Evelin A.; Coelho, Maria Alice Z.; Souza, Rodrigo O. M. A de; Simas, Alessandro B.C.; Freire, Denise M.G.

  PDF - p-61-61

• Abstract - Open Access

  Multicomponent Combinatorial Development of Prolyl Pseudo- Peptide Catalysts: Application in the Direct Asymmetric Michael Addition

  Torre, Alexander F. de la; Rivera, Daniel G.; Ferreira, Marco A. B.; Corrêa, Arlene G.; Paixão, Márcio W.

  PDF - p-62-62

• Abstract - Open Access

  New strategy for the synthesis of 4-amine-2-trifluoromethyl pyrroles N-substituted

  Aquino, Estefania da C.; Zanatta, Nilo; Gariboti, Vanessa C.; Bonacorso, Helio G.; Martins, Marcos A. P.

  PDF - p-63-63

• Abstract - Open Access

  Ultrasound-assisted synthesis of glycoporphyrin conjugates bearing carbamate and thiocarbamate linkers.

  Dallagnol, J. C. C.; Gonçalves, A. G.; Barreira, S. M. W.; Noseda, M. D.; Duarte, M. E. R.; Ducatti, D. R. B.

  PDF - p-64-64

• Abstract - Open Access

  NbCl5 as Catalyst in Diels-Alder Reaction of Furan Ring

  Santos, Deborah A. dos; Rodrigues, Ludmila R.; Jr., Valdemar Lacerda; Greco, Sandro J.; Neto, Alvaro C.; Santos, Reginaldo B. dos

  PDF - p-65-65

• Abstract - Open Access

  Application of a biarylarsine ligand in Heck and Stille reactions

  Quinteros, Gisela J.; Uberman, Paula M.; Martín, Sandra E.

  PDF - p-66-66

• Abstract - Open Access

  Facile one-pot synthesis of novel 1,2,4-Triazin-5-one from intramolecular cyclization

  Rosa, Fernanda A.; Gonçalves, Davana S.; Silva, Michael J. V. da; Tozatti, Camila S. S.; Gauze, Gisele F.

  PDF - p-67-67

• Abstract - Open Access

  Synthesis of Carbonohydrazideamide, Carbonohydrazidethioamide with potential biological activity

  Tozatti, Camila S. S.; Santos, Edson A. dos; Coelho, Narcimário P.; Santos, Maria Cristina P. dos; Silva, Michael J. V. da; Gonçalves, Davana S.; Basso, Ernani A.

  PDF - p-68-68

• Abstract - Open Access

  REACTIVITY STUDY OF METHYLCYCLOBUTYLKETONES AND CYCLOBUTANONES IN THE OBTENTION OF ANALOGS OF HYDANTOINIC NUCLEOSIDES

  Kuran, Juan A. Caturelli; Moglioni, Albertina G.

  PDF - p-69-69

• Abstract - Open Access

  1,3-Dipolar Cycloaddition Reactions of meso-Tetra(2’- thienyl)porphyrins with a Nitrile Oxide

  Momo, Patrícia B.; Ayres, Ricardo B.; Brocksom, Timothy J.; Oliveira, Kleber T. de

  PDF - p-70-70

• Abstract - Open Access

  Synthesis of some 1,2,3-triazole-chalcones as potential anticancer agents

  Pessôa, Jaqueline C.; Oliveira, Pãmella C. O. de; Fonseca, Meliza J. da C.; Pinheiro, Sergio; Muri, Estela M. F.; Dias, Ayres G.; Costa4, Paulo R. R.

  PDF - p-71-71

• Abstract - Open Access

  Asymmetrical Henry reaction using copper (II)/2-oxazoline complex.

  Mello, Murilo B. M.; Oliveira, Alfredo R. M.; Ribeiro, and Ronny R.

  PDF - p-72-72

• Abstract - Open Access

  Synthesis of meso-tetra-(5-iodo-thien-2-yl)-porphyrin; an intermediate for cross-coupling reactions

  Donatoni, Maria C.; Vieira, Ygor W.; Brocksom, Timothy J.; Oliveira, Kleber T. de

  PDF - p-73-73

• Abstract - Open Access

  Synthesis of novel amides derived from lumisantonin

  Moraes, Fernanda C.; Alvarenga, Elson S.; Amorim, Kariny B.

  PDF - p-74-74

• Abstract - Open Access

  Directed Functionalization of Quinoxalines Aiming the Synthesis of Bioactive Compounds

  Ferreira, Samuel R. A.; Pena, Jesus M.; Silva, Simone C.; Clososki, Giuliano C.

  PDF - p-75-75

• Abstract - Open Access

  3,4-(methylenodioxy)aniline as precursor to thiazolidinones

  Masteloto, Hellen G.; Drawanz, Bruna B.; Siqueira, Geonir M.; Cunico*, Wilson

  PDF - p-76-76

• Abstract - Open Access

  Enzymatic Kinetic Resolution of Hydroxy Furan and Tiophene 2-substituted

  Pires, D. S. F.; Ferreira, J. G.; Filho, E. F. S.; Princival, J. L.

  PDF - p-77-77

• Abstract - Open Access

  Studies aiming the synthesis of the indolizidine alkaloids (+)-Ipalbidine and (+)-Antofine

  Bertonha, Ariane F.; Burtoloso*, Antonio C. B.

  PDF - p-78-78

• Abstract - Open Access

  A Two-Step Synthesis of the Bioprotective Agent JP4-039 from N-Boc-L-Leucinal.

  Bernardim, Barbara; Burtoloso, Antonio C. B.

  PDF - p-79-79

• Abstract - Open Access

  Synthesis of (E)-1,2-bis-arylselanyl Alkenes Using Saccharomyces cerevisiae

  Lara, Renata G.; Soares, Liane K.; Santos, Juliana P.; Perin, Gelson; Lenardão, Eder J.; Vinueza., Julio C. G.

  PDF - p-80-80

• Abstract - Open Access

  Synthesis of new resorcinarene-based molecular clips

  Kvasnica, Miroslav; Purse, Byron W.

  PDF - p-81-81

• Abstract - Open Access

  Bioreduction of Alkynones by Fungus from Brazilian Northeast

  Silva, A. B. V.; Oliveira, J. R.; Ferreira, J. G.; Princival, J. L.; Nascimento, T. L.; Silva, D. C. V.; Souza, M. C.

  PDF - p-82-82

• Abstract - Open Access

  Total Synthesis and Revision of the Antidiabetic Activity of (-)-Tarchonanthuslactone

  Novaes, Luiz F. T.; Avila, Carolina M.; Souza, Gabriela F. P. de; Nascimento, Lucas F. R. do; Velloso, Licio A.; Pilli, Ronaldo A.

  PDF - p-83-83

• Abstract - Open Access

  New methodology of naphthoquinones esterification with longchain fat acids

  Gilles, V.; Vieira, A. M.; Lacerda Jr., V.; de Castro, E. V. R.; Greco, S. J.

  PDF - p-84-84

• Abstract - Open Access

  Electrophilic alkynylation of ketones using hypervalent iodine reagent: a new approach to quaternary carbon formation

  Utaka, Aline; Cavalcanti, Lívia N.; Jr., Luiz F. Silva

  PDF - p-85-85

• Abstract - Open Access

  Synthesis of all possible stereoisomers of 6,10,13- trimethyltetradecan-2-one, male-produced sex pheromone of Pallantia macunaima

  Soldi, Rafael A.; Zarbin, Paulo H.G.

  PDF - p-86-86

• Abstract - Open Access

  CARDANOL AND GLYCEROL AS BUILDING BLOCKS FOR THE SYNTHESIS OF NEW PORPHYRINS

  Souza, Daiane S.; Copini, Suély; Micheletti, Ana C.; Oliveira, Kléber T. de; Beatriz, Adilson

  PDF - p-87-87

• Abstract - Open Access

  Synthesis of Polyketide Fragments in Order to Study the Elaiophylin Biosynthesis

  Prediger, Patrícia; Dias., Luiz Carlos

  PDF - p-88-88

• Abstract - Open Access

  Virtual Screening of New Potential Organocatalysts for Stereoselective Nitroaldol Reactions

  Fernandes, Alessandra A. de G.; Papa, Bruna L.; Rodrigues, Alessandro

  PDF - p-89-89

• Abstract - Open Access

  Seleno-amino acid-based helical polymers for organocatalysis and functionalization of nanoparticles

  Gonçalves, A. C.; Dos Santos, A. A.

  PDF - p-90-90

• Abstract - Open Access

  New ESIPT fluorescent aldehydes as building blocks for organic photoactive compounds

  Affeldt, Ricardo F.; Santos, Fabiano da S.; Medeiros, Natália G.; Rodembusch, Fabiano S.

  PDF - p-91-91

• Abstract - Open Access

  Study of NH4[NbO(C2O4)2(H2O)].n H2O as a catalyst in transesterification of soybean oil to produce Biodiesel

  Arpini, Bruno Henrique; Sunderhus, Johann Castro Sodré; Jr., Valdemar Lacerda; Greco, Sandro José; Neto, Álvaro Cunha; Santos, Reginaldo Bezerra dos

  PDF - p-92-92

• Abstract - Open Access

  Studies on the synthesis of biodiesel catalyzed by Nb2O5.nH2O in transesterification reactions of cotton, coconut and flaxseed oils

  Sunderhus, Johann C. S.; Arpini, Bruno H.; Jr., Valdemar Lacerda; Greco, Sandro J.; Neto, Álvaro C.; Santos., Reginaldo B. dos

  PDF - p-93-93

• Abstract - Open Access

  Synthesis of selenium linked steroidal glycoconjugates

  Affeldt, Ricardo F.; Soares, Letiére C.; Rodrigues, Oscar E. D.; Ludtke, Diogo S.

  PDF - p-94-94

• Abstract - Open Access

  Synthesis of Optically Sugar Alcohols by Diastereoselective Addition of Organozinc Reagents

  Sachini, Maraisa; Lüdtke, Diogo S.

  PDF - p-95-95

• Abstract - Open Access

  Synthesis of New Triazoles by Click Chemistry

  Lima, Cíntia M. C. F.; Victor, Maurício M.; Rocha, Lenilson C.; Jeller, Alex H.; Porto, and André L. M.

  PDF - p-96-96

• Abstract - Open Access

  Synthesis of Substituted Pyrazolones from Morita-Baylis-Hillman Adducts

  Zeoly, Lucas A.; Barcelos, Rosimeire C.; Jr., Manoel T. Rodrigues; Martins, Lucimara J.; Coelho, Fernando

  PDF - p-97-97

• Abstract - Open Access

  Directed Magnesiation of Haloaromatic Oxazolines using the mixed lithium/magnesium base TMPMgCl.LiCl

  Batista, J.H.C.; Santos, F.M.; Silva, S.C.; Oliveira, A.R.M.; Clososki, G.C

  PDF - p-98-98

• Abstract - Open Access

  Synthesis of Chalcogenoacetylenes from Diorgano Diselenides and Terminal Acetylenes employing Bi (III)

  Souza, Matheus L.; Silva, Tiago L.; Rampon, Daniel S.; Rambo, Raoni S.; Radatz, Cátia S.; Schwab, Ricardo S.; Schneider*, Paulo H.

  PDF - p-99-99

• Abstract - Open Access

  Preliminary studies on Cu/SiO2 catalyzed imidazo[1,2-a]pyridine multicomponent synthesis

  Salles*, Helena D. de; Silva, Tiago L. da; Radatz, Cátia S.; Schneider, Paulo H.

  PDF - p-100-100

• Abstract - Open Access

  Synthesis of 3-hydroxy-2-(trimethylsilyl)phenyl trifluoromethanesulfonate as a versatile intermediate in preparative organic chemistry

  Moreira, Bárbara V.; Raminelli, Cristiano

  PDF - p-101-101

• Abstract - Open Access

  LDA Conjugate Addition to a Morita-Baylis-Hillman Ester: Experimental and DFT-based Theoretical Observations

  Sousa, Bruno A.; Paulino, Antonio A. S.; Braga, Ataualpa A. C.; Ando, Romulo A.; Santos, Alcindo A. Dos

  PDF - p-102-102

• Abstract - Open Access

  Synthesis of fused chromene-1,4-naphthoquionones under acid catalysis and microwave irradiation

  Rocha, David R. da; Mota, Kelly; Muniz, Illana; Ferreira, Vitor F.; Ferreira, Sabrina B.; Silva, Fernando de C. da

  PDF - p-103-103

• Abstract - Open Access

  Asymmetric enzymatic reduction and Suzuki-Miyaura coupling for the synthesis of odanacatib

  Lopes, Raquel de Oliveira; Reichart, Benedikt; Glasnov, Toma; Kappe, C. Oliver; Kroutil, Wolfgang; Miranda, Leandro Soter de M. e; Leal, Ivana Correa R.; Souza, Rodrigo O. M. A. de

  PDF - p-104-104

• Abstract - Open Access

  Three Step Chemo Enzymatic Continuous Flow Cascade Synthesis of 1-Monoacylglycerol.

  Itabaiana-Jr, Ivaldo; Souza, Rodrigo O. M. A. de

  PDF - p-105-105

• Abstract - Open Access

  Study toward the convergent total synthesis of the aporphine alkaloid PO-3

  Rossini, Allan F. C.; Raminelli, Cristiano

  PDF - p-106-106

• Abstract - Open Access

  Brønsted Acid Catalyzed Azlactone Ring Opening With a Wide Range Substratre Scope

  Pereira, Adriane A.; Castro, Pedro P. de; Mello, Amanda C. de; Amarante, Giovanni W.

  PDF - p-107-107

• Abstract - Open Access

  Brønsted Acid-Catalyzed Highly Diastereoselective Michaeltype Addition of Azlactones to Enones

  Ávila, Eloah P.; Mello, Amanda C. de; Diniz, Renata; Amarante, Giovanni W.

  PDF - p-108-108

• Abstract - Open Access

  Sugar-based Catalyst for the Highly Diastereoselective Desymmetrization of dbas

  Gonçalves, Jaqueline R.; Duarte, Talita N.; Pinheiro, Danielle L. J.; Amarante, Giovanni W.

  PDF - p-109-109

• Abstract - Open Access

  Synthesis of quinolines derivatives by multicomponent reaction promoted by NbCl5

  Santos, Giovanny Carvalho dos; Bartolomeu, Aloisio de Andrade; Silva-Filho., Luiz Carlos da

  PDF - p-110-110

• Abstract - Open Access

  Synthesis of new naphthotriazoles derived from juglone as anticancer agents

  Silva, Wanderson A. da; Moreira, Vinicius N.; Campos, Vinícius R.; Ferreira, Vitor F.; Rocha, David R. da; Resende, Jackson A. L. C.; Montenegro, Raquel C.; Souza, Maria Cecília B. V. de; Cunha, and Anna C.

  PDF - p-111-111

• Abstract - Open Access

  Study of the ortho-methoxy substituent group effect in selective demethylation reactions of methoxybenzoic acids.

  Gallo, Rafael D. C.; Alencar, Diandra P.; Yonekawa, Murilo; Muzzi, Rozanna M.

  PDF - p-112-112

• Abstract - Open Access

  Synthesis of 3-triazole-nor-β-lapachones with potential trypanocidal activity

  Cardoso, Mariana F. do Carmo; Rocha, David R. da; Salomão, Kelly; Castro, Solange de; Silva, Fernando de C. da; Ferreira, Vitor F.

  PDF - p-113-113

• Abstract - Open Access

  Study toward the total synthesis of lysicamine: an aporphine alkaloid with antileishmanial activity

  Muraca, Ana Carolina A.; Raminelli, Cristiano

  PDF - p-114-114

• Abstract - Open Access

  Microwave irradiation and DMC: a potent combination for the synthesis of 2-arylamino-3-tritylsulfanyl-propionic ethyl ester

  Santo, Stephanie Amarillis E.; Jr., Luiz S. Longo; Reis, Adriana Karla C. Amorim

  PDF - p-115-115

• Abstract - Open Access

  Reactions of bis-propargyl cycloalkanones with gold and silver catalysts

  Desiderá, André L.; Alves, Leandro de C.; Claro, Amanda M.; Domingos, Abner A.; Ferreira, Marco A. B.; Oliveira, Kleber T. de; Brocksom, Timothy J.

  PDF - p-116-116

• Abstract - Open Access

  Ring expansions of (R)-(–)-carvone to cycloheptenoid chirons

  Alves, Leandro de C.; Desiderá, André L.; Oliveira, Kleber T. de; Brocksom, Timothy J.

  PDF - p-117-117

• Abstract - Open Access

  Synthesis of 11a - Aza-5-deoxi-pterocarpans Via Palladium Aza-arylation of Dihydronaphtalen by Orto-iodoanilines Derivatives

  Buarque, Camilla D.; Fraga, Kevin C. de; Costa, Paulo R. R.

  PDF - p-118-118

• Abstract - Open Access

  Asymmetric Ring Contraction Reactions Mediated by Chiral I(III)

  Ahmad, Anees; Silva, Luiz F.; Jr.

  PDF - p-119-119

• Abstract - Open Access

  Novel Nano-Structured Chemosensors in Organic and Aqueous Phase

  Fernández-Lodeiro, Javier; Núñez, Cristina; Fernández-Lodeiro, Adrián; Oliveira, Elisabete; Santos, Hugo M.; Santos, Alcindo A. Dos; Capelo, José Luis; Lodeiro, Carlos

  PDF - p-120-120

• Abstract - Open Access

  New Emissive Rhodamine Dimer Probes for Mercury Detection in Solution, Gas Phase and Cellulose Supported Devices

  Núñez, Cristina; Bértolo, Emilia; Santos, Alcindo A. Dos; Diniz, Mario; Capelo, José Luis; Lodeiro, Carlos

  PDF - p-121-121

• Abstract - Open Access

  Targeting Echinococcus granulosus thioredoxin glutathione reductase using a Dynamic Combinatorial approach.

  Saiz, Cecilia; Castillo, Valerie; Salinas, Gustavo; Mahler., S. Graciela

  PDF - p-122-122

• Abstract - Open Access

  Efficient multicomponent synthesis of thiazolidinones from 2- aminoethyl(propyl)morpholine

  Gouvêa, Daniela Pires; Bervaldt, Gabriele dos Anjos; Neves, Adriana Machado das; Martins, Carolina; Cunico, Wilson João

  PDF - p-123-123

• Abstract - Open Access

  Chromenediones as potential plant growth regulators

  Alvarenga, Elson S.; Gomes, Maria Regina A.; Baia, Vitor C.; Souto, Francielly T.

  PDF - p-124-124

• Abstract - Open Access

  Synthetic Application of New Enaminodiketone: Regioespecific Synthesis of Aza-Heterocycles

  Rosa, Fernanda A.; Silva, Michael J. V. da; Gonçalves, Davana S.; Arita, Daniela H.; Tozatti, Camila S. S.; Bandoch, Gisele de F. G.

  PDF - p-125-125

• Abstract - Open Access

  Synthesis of new heterocyclic isosteres of L-buthionine sulfoximine (L-BSO)

  P., Thomas; R., Armijo; A., Tapia R.; C., Salas

  PDF - p-126-126

• Abstract - Open Access

  Ni-Catalyzed Silylation of Inert C-O Bonds under Mild Conditions

  Zárate, Cayetana; Martin, Rubén

  PDF - p-127-127

• Abstract - Open Access

  Efficient Asymmetric Synthesis of Lamivudine and its enantiomer via Enzymatic Dynamic Kinetic Resolution

  Hu, Lei; Schaufelberger, Fredrik; Zhang, Yan; Ramström, Olof

  PDF - p-128-128

• Abstract - Open Access

  Selective semi-synthesis of dihydrocucurbitacin B glycosides

  MOROTTI, A. L. M.; ZIMMERMANN, L. A.; MACHADO, V. R.; SCHENKEL, E. P.; BERNARDES, L. S. C.

  PDF - p-129-129

• Abstract - Open Access

  Asymmetric synthesis of pyranocumarins under greener conditions

  Monteiro, J. L.; Torre, A. F.; Paixão, M. P.; Corrêa, A. G.

  PDF - p-130-130

• Abstract - Open Access

  Synthesis of new ionophilic SNS ligands and their Ru(II) complexes

  Matiello, Gabriela I.; Dupont, Jairton; Ebeling, Günter

  PDF - p-131-131

• Abstract - Open Access

  Binding site elucidation of a small molecule inhibitor of FtsZ

  Nepomuceno, Gabriella M.; Anderson, David E.; Tadeus, Clarissa; Wang, Qian; Painter, Phillip P.; Chan, Katie M.; O’Brien, Terrence E.; Sarabia, Francisco J.; Tantillo, Dean J.; Ames, James B.; Lebrilla, Carlito; Shaw, Jared T.

  PDF - p-132-132

• Abstract - Open Access

  Synthesis of chiral 4-pyrazolyl dihydropyridines and their enantiomeric separation

  Kumar, Rakesh; Yadav, Neha; Arora, Jyoti; Prasad, Ashok K

  PDF - p-133-133

• Abstract - Open Access

  Studies of continuous-flow synthesis of nonpeptidal bistetrahydrofuran moiety of Darunavir

  Leão, Raquel A. C.; Gosmann, Grace; Muniz, Mauro N.; Miranda, Leandro S. de M. e; Souza, Rodrigo O. M. A. de

  PDF - p-134-134

• Abstract - Open Access

  Strategies for Total Synthesis of Pyrenophorin

  Barbosa, Jaqueline Rosa C.; Victor, Mauricio Moraes

  PDF - p-135-135

• Abstract - Open Access

  SYNTHESIS OF A NEW CHIRAL BIS-ARSINE LIGAND BASED ON NATURAL CARBOHYDRATES

  Puenzo, Sol C. Parajón; Badano, Joaquín Arata; Vidal, Martin G. Lopez; Varela, Oscar; Martín, Sandra E.

  PDF - p-136-136

• Abstract - Open Access

  Discovery and synthesis of a new analogues of the cyclopenta[b]indoles as tubulin polymerization inhibitors

  Fernandes, D. C.; Santos, R. N. S.; Júnior, M. T. R; Andricopulo, A. D.; Coelho, F.

  PDF - p-137-137

• Abstract - Open Access

  Stereoselective hydrogenation of 3-acyl-substituted 2- (trifluoromethyl)-2H-chromen-5-one and chromane scaffolds in NaBH4 /ethanol medium

  Navarini, Jussara; (PQ), Helio G. Bonacorso; Wiethan, Carson W.; Pittaluga, Everton P.; Junges, Andrizia F.; Luz, Fábio M.; Martins, Marcos A. P.; Zanatta, Nilo

  PDF - p-138-138

• Abstract - Open Access

  Theoretical study of the regiospecific synthesis of pyrazole-5- carboxylate from unsymmetrical enaminodiketones

  Rozada, Thiago C.; Silva, Michael J. V. da; Pontes, Rodrigo M.; Basso, Ernani A.; Rosa, Fernanda A.

  PDF - p-139-139

• Abstract - Open Access

  Benzo[b]thiophene dimerization: A promising experimental finding directed to the C-3 functionalization with aryl alcohols.

  Romero-Parra, Javier; Pessoa-Mahana, Hernán; Pessoa-Mahana., C. David

  PDF - p-140-140

• Abstract - Open Access

  SINTHESYS OF CINNAMIC ACID DERIVATIVES WITH CORROSION INHIBITION ACTIVITY FOR CARBON STEEL ALLOY

  VIANA, Thiago Silva; DUQUE, Pedro Henrique Fonseca; PINTO, Camila Prestes; AGUIAR, Ana Luiza Carvalho Guimaraes; SOUZA, Flávia Carvalho; COTRIM, Bruno Almeida; RESENDE, Gabriel de Oliveira; BARRETO JR, Cleber Bomfim

  PDF - p-141-141

• Abstract - Open Access

  New 1,3,4-Oxadiazolyl-pyrazolyl-Pyridine Tricyclic Scaffold Derivatives: Synthesis and Structure Assignment by NMR and DFT Calculations

  Paim, Gisele R.; Meira, Susiane C.; Pittaluga, Everton P.; Porte, Liliane M. F.; Meyer, Alexandre R.; Navarini, Jussara; Bonacorso, Helio G.

  PDF - p-142-142

• Abstract - Open Access

  Aluminum promotes easy access to high substituted trihalomethyl triazolyl homoallylic alcohols

  Wiethan, Carson W.; Bonacorso, Helio G.; Moraes, Maiara C.; Andrighetto, Rosália; Belo, Chaiene R.; Martins, Marcos A. P.; Zanatta, Nilo

  PDF - p-143-143

• Abstract - Open Access

  Cu-catalyzed Mild C(sp2)-H Functionalization Assisted by Carboxylic Acids En Route to Hydroxylated Arenes

  Gallardo-Donaire, Joan; Martin, Ruben

  PDF - p-144-144

• Abstract - Open Access

  Synthesis of two new series of 7-aminocarbohydrateisoquinoline- 5,8-dione derivatives

  Silva, Wanderson A. da; Santos, Angela Cristina P. B. dos; Ferreira, Vitor F.; Montenegro, Raquel C.; Campos, Vinícius R.; Souza, Maria C. B. V. de; Cunha, Anna C.

  PDF - p-145-145

• Abstract - Open Access

  Ritter reaction of N-(hydroxymethyl)saccharin with nitriles: synthesis of new N-(amidomethyl)saccharins

  Mattos, Marllon N. de Oliveira e Marcio C. S. de

  PDF - p-146-146

• Abstract - Open Access

  Influence of the Phenylsulfonylethylidene (PSE) Acetal Clamp on the Glycosylation Involving Thioglycoside Donors

  Oliveira, Ronaldo N. de; Schuler, Marie; *, Arnaud Tatibouët; Rollin, Patrick

  PDF - p-147-147

• Abstract - Open Access

  General substrates for stereoselective synthesis: utilization of D- and L-arabinose

  Soares, Fábio da Paixão; Silva, Maria Joselice e; Doboszewski, Bogdan

  PDF - p-148-148

• Abstract - Open Access

  C5 atom of D-galactopyranose as a source of chirality: preliminary results

  Silva, Maria Joselice e; Silva, Paulo Roberto da; Doboszewski, Bogdan

  PDF - p-149-149

• Abstract - Open Access

  Synthesis of Quinoline-Triazoil Carboxylates by Organocatalytic Cycloaddition of β-Ketoesters and 4-Azido-7-Chloroquinoline

  Saraiva, Maiara; Krüger, Roberta; Alves, Diego

  PDF - p-150-150

• Abstract - Open Access

  Towards the synthesis of 27-Deoxylyngbyabellin A analogues as potential chemotherapeutics.

  Scarone, Laura; Sandin, Leonardo; Serra., Gloria

  PDF - p-151-151

• Abstract - Open Access

  First Total Synthesis of Aerucyclamide B and Macrocycle Analogs as Antimalarial and Anti-Trypanosomal Agents

  Peña, S.; Scarone, L.; Medeiros, A.; Comini, M.; Stewart, L.; Yardley, V.; Albericio, F.; Serra, G.

  PDF - p-152-152

• Abstract - Open Access

  Acetonides as Masked Nucleophiles in the Gold-Catalyzed Spiroketalization of Monopropargylic Triols.

  Paioti, Paulo H. S.; Ketcham, John M.; Aponick, Aaron

  PDF - p-153-153

• Abstract - Open Access

  Synthesis of lactones and lactams analogues to rubrolides as inhibitors of Enterococcus faecalis biofilm formation

  Pereira, Ulisses A.; Barbosa, Luiz C. A.; Maltha, Célia R. A.; Demuner, Antônio Jacinto; Pimenta, Andréa de L.

  PDF - p-154-154

• Abstract - Open Access

  Metal-Free sp2 and sp3 C-H Functionalization/C-O Bond Forming Reaction

  Wang, Xueqiang; Donaire, Joan G.; Martin, Ruben

  PDF - p-155-155

• Abstract - Open Access

  Synthesis of novel [2]rotaxanes using hydrogen-bonding template

  Rodrigues, Letícia V.; Buriol, Lilian; Frizzo, Clarissa P.; Berná, José; Alajarín, Mateo; Martins, Marcos A. P.

  PDF - p-156-156

• Abstract - Open Access

  A New Approach to Atropisomerism

  Cardoso, Flávio Sêga Pereira; Aponick, Aaron

  PDF - p-157-157

• Abstract - Open Access

  Povarov reaction for the synthesis of 2-(2-pyridyl)quinoline

  Barbosa, Luiz C. A.; Borel, Carmindo R.; Fernandes, Sergio A.; Maltha, Célia R. A.

  PDF - p-158-158

• Abstract - Open Access

  Synthesis of β-enaminones catalyzed by nanoparticles of Fe2O3 in ultrasound and solvent-free approach.

  Hortelan, Cristiane Regina Winck; Silveira, Ingridhy Ostaciana Maia Freitas da; Souza, Silvia Mendes de; Beatriz, Adilson; Gomes, Roberto da Silva; Domingues, Nelson Luís de Campos

  PDF - p-159-159

• Abstract - Open Access

  Coumarins from Free ortho-Hydroxy Cinnamates by Heck- Matsuda Arylations and their Application in the Total Synthesis of (R)-Tolterodine

  Barancelli, Daniela Aline; Jr., Airton G. Salles; Taylor, Jason G.; Correia, Carlos Roque D.

  PDF - p-160-160

• Abstract - Open Access

  Oxireduction’s Studies of Arytetralone and Aryltetralol Mediated by Rhodotorula sp

  Capeletto, Marina G.; Jr, Luiz S. Longo; Batista, Wagner L.; Bianco, Graziela G.

  PDF - p-161-161

• Abstract - Open Access

  Construction of Diarylmethane Compounds. Synthesis of tolpropamine via Heck-Matsuda Reaction

  Silva, Allan Ribeiro da; Prediger, Patrícia; Correia, Carlos Roque Duarte

  PDF - p-162-162

• Abstract - Open Access

  Studies toward total synthesis of tautomycetin

  Sant’Ana, Danilo P.; Fiqueiredo, Renata Marcia de; Campagne, Jean-Marc; Dias., Luiz Carlos

  PDF - p-163-163

• Abstract - Open Access

  Coumarins and Neoflavones: Synthesis and HCV NS5B Polymerase Inhibition

  Moraes, Paula de F. de; Leão, Raquel A. C.; Nichols, Daniel Brian; Basu, Amartya; Chudayeu, Maksim; Talele, Tanaji T.; Kaushik-Basu, Neerja; Costa, Paulo R. R.

  PDF - p-164-164

• Abstract - Open Access

  Synthesis of ligands for nuclear receptors of thyroid hormones

  Castro, Guilherme V. de; Sanches, Vitor Lacerda; Donate, Paulo M.; Polikarpov, Igor; Sairre, Mirela I. de

  PDF - p-165-165

• Abstract - Open Access

  p-Sulfonic acid calix[4]arene as a new reusable organocatalyst for the transesterification of vegetable oil

  Almeida, Camila Guimarães de; Souza, Isabella Flores de; Fernandes, Sergio Antônio; Hyaric, Mireille Le

  PDF - p-166-166

• Abstract - Open Access

  The oxidation of indole derivatives using dimethyl dioxirane

  Marçal*, Luisa L.; Garden, Simon J.

  PDF - p-167-167

• Abstract - Open Access

  Benzocarbazolquinones and Benzonaphthofurandiones by Palladium Catalyzed Oxidative C-H Functionalization

  Lisboa, Cinthia da Silva; Santos, Gustavo dos; Lucas, Nanci C. de; Garden, Simon J.

  PDF - p-168-168

• Abstract - Open Access

  Highly regioselective epoxide hydrogenolysis aiming at the bulgecinine synthesis

  Martinez, Pablo David G.; Correia, Carlos Roque D.

  PDF - p-169-169

• Abstract - Open Access

  Synthesis of new N-confused triazole-porphyrin derivatives through the Heck procedure

  Gomes, Ana T.P.C.; Silva, Fernando C. da; Neves, Maria G.P.M.S.; Ferreira, Vítor F.; Cavaleiro, José A. S.

  PDF - p-170-170

• Abstract - Open Access

  Phenanthridine derivatives via palladium catalyzed intramolecular functionalization of C(sp2)-H bonds.

  Costa, Roberta L. da; Garden, Simon J.

  PDF - p-171-171

• Abstract - Open Access

  Synthesis of 2,5-disubstituted selenazoles by O-Se exchange

  Pizzo, Chiara; Mahler, Graciela

  PDF - p-172-172

• Abstract - Open Access

  Syntheses of β-hydroxy-α-amino esters and non-proteinogenic α-amino acids from Morita-Baylis-Hillman adducts.

  Ullah, Hamid; Ferreira, Andre V.; Jr, Manoel T. Rodrigues; Coelho, Fernando

  PDF - p-173-173

• Abstract - Open Access

  Synthesis and characterization of novel phosphinamide bidentate ligands with groups P=O, P=S and P=Se: Application in coordination chemistry with Zn++

  Bastos, Neidemar de M. S.; Macedo, Júlia T. de; Souza, Marcos C. de; Romeiro, Gilberto A.; Resende, Jackson A. L.C.; Iglesias, María J.; Ortiz, Fernando L.; Casimiro, María; Freitas., Maria C. R.

  PDF - p-174-174

• Abstract - Open Access

  Studies on the synthesis of (poly)arylacetylenes using cardanol and glycerol as raw materials

  Matayoshi, Tatiana; Micheletti, Ana Camila; Beatriz, Adilson

  PDF - p-175-175

• Abstract - Open Access

  Synthesis of 7-trifluo[trichlo]romethyl-5-aryl[alkyl]-tetrazolo[1,5-a] pyrimidines in Ionic Liquid

  Scapin, Elisandra; Buriol, Lilian; Frizzo, Clarissa Piccinin; Martins, Marcos A. P.

  PDF - p-176-176

• Abstract - Open Access

  A versatile synthesis to trisubstituted nitroalkenes via nitroaldol reaction: Synthesis of Baylis-Hillman type adducts

  Pereira, Vera L. Patrocinio; Costa, Jeronimo da Silva; Silva, Alessandra C. de Souza e; Nascimento., Fernanda Cunha do

  PDF - p-177-177

• Abstract - Open Access

  Synthesis of glycopeptides mimetics of T. cruzi and tumor mucins as potential vaccines

  Campo, Vanessa Leiria; Baruffi, Marcelo Dias; Carvalho, Ivone

  PDF - p-178-178

• Abstract - Open Access

  Intramolecular Aza-Anti-Michael Addition for the Synthesis of 2-Iminothiazolidines

  Ferreira*, Misael; Sá, Marcus Mandolesi

  PDF - p-179-179

• Abstract - Open Access

  Synthesis of novel phosphinamide phosphoramidate conjugates with possible applications in catalysis

  Medeiros, Antonia Carlene R. F.; Bernardino, Alice Maria R.; Souza, Marcos C. de; Ortiz, Fernando L.

  PDF - p-180-180

• Abstract - Open Access

  Regioselective reduction of 1-amino-2,4-dinitrobenzenes

  Custódio, Cíntia de Andrade; Garden, Simon J.

  PDF - p-181-181

• Abstract - Open Access

  Synthesis of novel 6-seleno-dihydropyrimidinones: Potentially bioactive compounds

  Barbosa, Flavio A. R.; Canto, Rômulo F. S.; Braga, Antonio L.

  PDF - p-182-182

• Abstract - Open Access

  Synthesis of Thiophene Acetylenes via Sonogashira Cross- Coupling Reactions

  Carvalho, Diego B.; Andrade, Camila B.; Miranda, Carla R. Z.; Hurtado, Gabriela R.; Viana, Luiz H.; Jr., Palimécio G. Guerrero; Baroni, Adriano C. M.

  PDF - p-183-183

• Abstract - Open Access

  Microwave-assisted synthesis and antifungal activity of calix[4]aldimines

  Silva, Cleiton M. da; Magalhães, Thais F.F.; Silva, Danielle L. da; Alves, Rosemeire B.; Resende-Stoianoff, Maria A. de; Fátima, Ângelo de

  PDF - p-184-184

• Abstract - Open Access

  α-Hydroxylation of malonates under mild reaction conditions

  Peterle, Marcos M.; Marques, Marcelo V.; Sá, Marcus M.

  PDF - p-185-185

• Abstract - Open Access

  Diastereoselective synthesis of dihydroquinolines and tetrahydroquinolines from Morita Baylis-Hillman adducts

  Jr., Manoel T. Rodrigues; Agy, Andre Capretz; Lustosa, Danilo Machado; Coelho, Fernando

  PDF - p-186-186

• Abstract - Open Access

  New Aza-pterocarpan Analogues by Intramolecular 1,3-Dipolar Cycloaddition in in situ generated nitroneolefins

  Barcellos, Julio C. F.; Dias, Ayres G.; Costa, Paulo R. R.

  PDF - p-187-187

• Abstract - Open Access

  Studies on the enantioselective Heck arylation of Ncarboethoxy 3-pyrroline with aryldiazonium salts

  Lustosa, Danilo Machado; Correia, Carlos Roque D.

  PDF - p-188-188

• Abstract - Open Access

  Stereoselective Synthesis of Divinylic Chalcogenides Using PEG-400

  Soares, Liane K.; Luz, Eduardo Q.; Webber, Rodrigo; Borges, Elton L.; Perin., Gelson

  PDF - p-189-189

• Abstract - Open Access

  An expeditious approach to (+)-polyoxamic acid and derivatives from asymmetric Morita-Baylis-Hillman reaction.

  Guidotti, Bruno Boni; Correia, José Tiago Menezes; Ullah, Hamid; Coelho., Fernando Antônio Santos

  PDF - p-190-190

• Abstract - Open Access

  PEG: An Efficient Green Solvent for Organocatalytic Asymmetric Michael Addition

  Feu, Karla S.; Silva, Sandrina I. R. M.; Junior, Marco A. F. M.; Torre, Alexander F. de la; Corrêa, Arlene G.; Paixão, Márcio W.

  PDF - p-191-191

• Abstract - Open Access

  Synthesis of oxirane from quinones against T. cruzi

  Carneiro, Paula F.; Rocha, Alice S.B.; Lechuga, Guilherme C.; Nascimento, Samara B.; Pinto, Maria do Carmo F.R.; Bourguignon, Saulo C.; Ferreira, Vitor F.

  PDF - p-192-192

• Abstract - Open Access

  Synthesis of novel Imidazolidinone Peptidomimetics

  Krake, Susann H.; Bergmeier, Stephen C.

  PDF - p-193-193

• Abstract - Open Access

  Synthesis of a new class of 2-bromo-3-amino-1,4- naphthoquinone glycoconjugates

  Dias, Flaviana Rodrigues Fintelman; Ferreira, Vitor Francisco; Campos, Vinícius Rangel; Montenegro, Raquel C.; Souza, Maria Cecília B. V. de; Cunha, Anna Claudia

  PDF - p-194-194

• Abstract - Open Access

  Multicomponent synthesis of R-(+)-limonene-based 1,3,4-thiadiazoles

  Falzirolli, Hugo; Vandresen, Fábio; Furlan, Francieli; Silva., Cleuza Conceição da

  PDF - p-195-195

• Abstract - Open Access

  Synthesis of Diselenide Based Picolylamide Derivatives: Biologically Potential Compounds

  Rafique, Jamal; Saba, Sumbal; Canto, Rômulo F. S.; Hassan, Waseem; Rocha, João B. T.; Braga, Antonio L.

  PDF - p-196-196

• Abstract - Open Access

  Synthesis of New Diselenide Based Ester Derivatives: Biologically Potential Compounds

  Saba, Sumbal; Rafique, Jamal; Godoi, Marcelo; Hassan, Waseem; Rocha, João Batista T.; Braga, Antonio L.

  PDF - p-197-197

• Abstract - Open Access

  Solid Phase Synthesis of Hexapeptides and Solution Macrocyclization to Obtain Antiparasitic Agents

  Fagundez, Catherine; Sellanes, Diver; Medeiros, Andrea; Comini, Marcelo; Stewart, Lindsay; Yardley, Vanessa; Serra, Gloria

  PDF - p-198-198

• Abstract - Open Access

  Reaction of vinylbromides with alkynes using ppm amounts of Pd as catalyst

  Biajoli*, André F. P.; Monteiro, Adriano L.

  PDF - p-199-199

• Abstract - Open Access

  Synthesis and development of novel small molecules targeting Rac1 signaling as new potential leads for antitumor agents

  Ciarlantini, M.; Gonzalez, N; Cardama, G. A.; Defelipe, L.; Turjanski, A.; Alonso, D. F.; Gomez, D. E.; Lorenzano Menna, P.; Comin, M. J.

  PDF - p-200-200

• Abstract - Open Access

  Synthesis and photophysical properties of a Tröger’s basetriazole- linked glycoconjugate

  Pimentel, Débora M.; Vargas, Jaqueline P.; Lüdtke, Diogo S.; Rodembusch, Fabiano S.

  PDF - p-201-201

• Abstract - Open Access

  Organocatalytic Michael reaction study between phenyl acetaldehyde and nitrostyrene

  Gandolfi Donadío, Lucía; Galetti, Mariana A.; Giorgi, Gianluca; Comin, Maria J.

  PDF - p-202-202

• Abstract - Open Access

  Coibacins A and B: Total Synthesis, Stereochemical Revision and Structural Elucidation

  Avila, Carolina M.; Carneiro, Vânia M. T.; Balunas, Marcy J.; Gerwick, William H.; Pilli, Ronaldo A.

  PDF - p-203-203

• Abstract - Open Access

  β-C-ribosyl-1,2,3-triazole analogues of guanosine as potencial antiviral agents against dengue and hepatitis C virus

  Lopes, Alexandra Basilio; Romeiro, Nelilma Correia; Tanuri≠, Amilcar; Germain, Nadège Lubin-; Souza, Rodrigo Octávio M. A. de; Miranda, Leandro S.M.

  PDF - p-204-204

• Abstract - Open Access

  Synthesis of isobenzofuranones by Diels-Alder reaction

  Teixeira, Milena G.; Alvarenga, Elson S.; Demuner, Antonio J.; Maltha, Célia R. A.; Barbosa, Luiz Claudio A.

  PDF - p-205-205

• Abstract - Open Access

  Synthesis of trifluoromethyl benzamides and their effects on the photosynthetic machinery

  Teixeira, Róbson Ricardo; Bressan, Gustavo Costa; Barros, Marcus Vinícius de Andrade; Forlani, and Giuseppe

  PDF - p-206-206

• Abstract - Open Access

  Cross-coupling reactions as a strategy for Naphthalocyanine synthesis

  Gobo, Nicholas R. S.; Brocksom, Timothy J.; Oliveira, Kleber T. de

  PDF - p-207-207

• Abstract - Open Access

  Determination of the absolute configuration of 6 -Hydroxitricyclo[ 6.2.1.02,7]undeca-9-ene-3-one by chemical correlation

  Ito, Felícia Megumi; Copini, Suély; Almeida, Nathália Rodrigues de; Pedroni, Kelly Karoliny Lima; Micheletti, Ana Camila; Beatriz, Adilson

  PDF - p-208-208

• Abstract - Open Access

  Immobilization of CuSO4 on alginate for synthesis of α- triazoloketones

  Silva, Natália A. da; Ferreira, Irlon M.; Porto, André Luiz M.

  PDF - p-209-209

• Abstract - Open Access

  Semi-synthesis of Purpurinimides: The search for more effective PDT agents

  Uliana, Marciana P.; Brocksom, Timothy J.; Oliveira, Kleber T. de; Bagnato, Vanderlei S.; Kurachi., Cristina

  PDF - p-210-210

• Abstract - Open Access

  Synthesis and photophysical properties of 2,5-diarylindolizines

  Souza, Camila R.; Amaral, Mônica F. Z. J.; Clososki, Giuliano C.

  PDF - p-211-211

• Abstract - Open Access

  Synthesis of meso-N-Phenylmaleimide-porphyrins

  Santos, Fabiane A. B. dos; Carvalho, Carla M. B.; Santos, Edjane R. dos; Brocksom, Timothy J.; Oliveira, Kleber T. de

  PDF - p-212-212

• Abstract - Open Access

  Effects on Circular Dicroism of pyridil-oxazolinic monomers: preparatory studies on the helical polymer synthesis

  Sakae, George H.; Carmona, Rafaela C.; Wendler, Edison P.; Santos, Alcindo A. Dos

  PDF - p-213-213

• Abstract - Open Access

  A high enantioselective Proline-based helical polymer catalyst for aldol type reaction

  Sakae, George H.; Takata, Leandro M.; Paulino, Antonio S.; Bazito, Reinaldo C.; Cassaro, Rafael F.; Princival, Cleverson; Santos, Alcindo A. Dos

  PDF - p-214-214

• Abstract - Open Access

  1,3-Dipolar cycloadditions for the synthesis of low aggregation chlorins: A methodological study

  Souza, Juliana M. de; Assis, Francisco F. de; Carvalho, Carla M. B.; Cavaleiro, José A. S.; Brocksom, Timothy J.; Oliveira, Kleber T. de

  PDF - p-215-215

• Abstract - Open Access

  Organocatalysis in the Three-Component Povarov Reaction and Mechanistic Investigation by Mass Spectrometry

  Simões, Juliana B.; Fátima, Ângelo de; Sabino, Adão A.; Aquino, Francisco J. T.; Silva, Daniel L.; Barbosa, Luiz Claudio A.; Fernandes, Sergio A.

  PDF - p-216-216

• Abstract - Open Access

  Base/Electrophile-Controlled Regioselective Functionalization of 1-Substituted-Indolizines

  Amaral, Mônica F. Z. J.; Baumgartner, Amanda A.; Clososki, Giuliano C.

  PDF - p-217-217

• Abstract - Open Access

  Synthesis and photophysical evaluations of β-fused Uracil- Porphyrin derivatives

  Fujita, Marta Akemi; Carvalho, Carla Marisa Brito; Brocksom, Timothy John; Oliveira, Kleber Thiago de

  PDF - p-218-218

• Abstract - Open Access

  Synthetic studies for bisthiazolidine stepwise preparation

  Castillo, Valerie; Mahler, Graciela

  PDF - p-219-219

• Abstract - Open Access

  Synthesis and photophysical studies of a chlorin sterically designed to prevent self-aggregation

  Assis, Francisco F. de; Souza, Juliana M. de; Assis, Beatriz H. K.; Brocksom, Timothy J.; Oliveira, Kleber T. de

  PDF - p-220-220

• Abstract - Open Access

  Synthesis of 3,4-dibromo-1H-pyrrole-2-carbaldehyde: a building block for preparation of tetrabromobacteriochlorins

  Assis, Francisco F. de; Brocksom, Timothy J.; Oliveira., Kleber T. de

  PDF - p-221-221

• Abstract - Open Access

  Total Synthesis of Isoellipticine

  Naciuk, Fabrício Fredo; Malanzuk, Rebeca; Fontoura, Luiz Antonio Mazzini; Miranda, Paulo C. M. L.

  PDF - p-222-222

• Abstract - Open Access

  Synthesis and antitumor activity of novel Schiff bases derived from 6-hydroxy-1,3-benzoxathiol-2-one

  Chazin, Eliza de L.; Sanches, Paola de S.; Júnior, Walcimar T. Vellasco; Gomes, Claudia R. B.; Montenegro, Raquel C.; Vasconcelos, Thatyana R. A.

  PDF - p-223-223

• Abstract - Open Access

  Synthesis of news furo[2,3-d] pyrimidine derivatives as potential inhibitors of DHFR

  Ferreira, Marcelle de Souza; Villar, José Daniel Figueroa

  PDF - p-224-224

• Abstract - Open Access

  Michael type reactions mediated by NbCl5.

  Rodrigues*, Shirley Muniz Machado; Silva., Gil Valdo José da

  PDF - p-225-225

• Abstract - Open Access

  NANOASSEMBLIES: COVALENT DERIVATIVES OF NEVIRAPINE WITH POLYETHYNE GLYCOL DIACRYLATE

  E, Costas do Santos; R., Glisoni; L., Fabian; A., Sosnik; A., Moglioni

  PDF - p-226-226

• Abstract - Open Access

  Synthesis of polisubstituted 1,3-azadienes from enaminones

  Marques, Monique F.; Cunha, Silvio

  PDF - p-227-227

• Abstract - Open Access

  Studies on the Regio- and Enantioselective Heck Arylations of Acyclic Allylic Alcohols.

  Oliveira, Caio C.; Correia, Carlos Roque D.

  PDF - p-228-228

• Abstract - Open Access

  Microwave induced multicomponent synthesis of 2-pyrrolo-3’-yloxindoles through reaction of enaminone, isatin and phosphorus ylide

  Cunha, Silvio; Filho, Raimundo Francisco dos Santos

  PDF - p-229-229

• Abstract - Open Access

  Studies Towards Asymmetric Total Synthesis of Populene D

  Ishikawa, Eloisa E.; Jr., Luiz F. Silva

  PDF - p-230-230

• Abstract - Open Access

  P,S-ligands for Ir-catalyzed Asymmetric Hydrogenation of Minimally Functionalized Olefins – A Theoretical Study

  Karlsson, Erik A.; Margalef, Jèssica; Mazuela, Javier; Pàmies, Òscar; Diéguez, Montserrat; Pericàs, Miquel A.

  PDF - p-231-231

• Abstract - Open Access

  The Diels-Alder reaction of para-benzoquinones and simple dienes under catalysis with FeCl3 on Aerosil® silica

  Donatoni, Maria C.; Junior, Gilmar A. B.; Santos, Alcindo A. Dos; Oliveira, Kleber T. de; Brocksom, Timothy J.

  PDF - p-232-232

• Abstract - Open Access

  Study toward the synthesis of (R)-(-)-aporphine

  Perecim, Givago P.; Raminelli, Cristiano

  PDF - p-233-233

• Abstract - Open Access

  Ultrasonics promoted synthesis of thiazolidinones from 2- aminopyridine

  Bosenbecker, Juliano; Gouvêa, Daniela P.; Siqueira, Geonir M.; Cunico, Wilson

  PDF - p-234-234

• Abstract - Open Access

  Cyclization of Homoallylic Alcohols with Iodine/Iodine(III)

  Scarassati, Paulo; Jr., Luiz F. Silva

  PDF - p-235-235

• Abstract - Open Access

  Gold-Catalyzed Cyclization of Ynamides and Propargylic Carboxylates

  Wieteck, Marcel; Rettenmeier, Eva; Hashmi, A. Stephen K.

  PDF - p-236-236

• Abstract - Open Access

  Preparation of New Magnesium Carbenoids Aiming Inhibitors of HIV-1 Protease Synthesis

  Nishimura, R. H. V.; Toledo, F. T.; Clososki, G. C.

  PDF - p-237-237

• Abstract - Open Access

  Study on the intermolecular Enantioselective Heck-Matsuda reaction of acyclic olefin diol

  Frota, Carlise; Oliveira, Caio Costa; Correia., Carlos R. D.

  PDF - p-238-238

• Abstract - Open Access

  Glyco-Porphyrins and -Phthalocyanines for Cancer Photodynamic Therapy

  Pereira, Patrícia M. R.; Lourenço, Leandro M. O.; Bispo, Mafalda A. F.; Silva, Sandrina; Cavaleiro, José A. S.; Ribeiro, Carlos A. F.; Fernandes, Rosa; Tomé, João P. C.

  PDF - p-239-239

• Abstract - Open Access

  Nickel-Catalyzed Borylation of Halides and Pseudohalides with Tetrahydroxydiboron [B2(OH)4]1

  Cavalcanti*, Livia N.; Molander, Gary A.

  PDF - p-240-240

• Abstract - Open Access

  Synthesis of New Mitotane Analogues

  Santana, Amanda S.; Sampaio, Felipe R.; Correia, Carlos Roque D.

  PDF - p-241-241

• Abstract - Open Access

  Chemoenzymatic synthesis of derivatives azoles by lipase from Pseudomonas fluorescens

  Ferreira, Irlon M.; Porto, André L. M.

  PDF - p-242-242

• Abstract - Open Access

  Integrated Batch and Continuous Flow Process for the Synthesis of Goniothalamin

  Pastre, Julio C.; Murray, Philip R. D.; Browne, Duncan L.; Pilli1, Ronaldo A.; Ley, Steven V.

  PDF - p-243-243

• Abstract - Open Access

  Continuous Flow-Processing of Organometallic Reagents Using an Advanced Peristaltic Pumping System and the Telescoped Flow Synthesis of (E/Z)-Tamoxifen

  Murray, Philip R. D.; Browne, Duncan L.; Pastre, Julio C.; Ley, Steven V.

  PDF - p-244-244

• Abstract - Open Access

  Microwave-assisted Synthesis of New Ethyl 2-aminopyrimidine- 4-carboxylates

  Vargas, Pâmela S. de; Bonacorso, Helio G.; Zanatta, Nilo; Frizzo, Clarissa P.; Martins, Marcos A. P.

  PDF - p-245-245

• Abstract - Open Access

  Sonochemistry to promote the synthesis of 5- arilydenethiazolidine-2,4-diones

  Drawanz, Bruna Bento; Ribeiro, Camila; Masteloto, Hellen G.; Cunico, Geonir M. Siqueira Wilson

  PDF - p-246-246

• Abstract - Open Access

  Glycerol as solvent to the synthesis of thiazolidinones

  Bervaldt, Gabriele dos Anjos; Gouvêa, Daniela Pires; Neves, Adriana Machado das; Difabio, Roberta; Cunico, Wilson João

  PDF - p-247-247

• Abstract - Open Access

  Enantioselective Arylation of Aliphatic Aldehydes Catalyzed by Chiral Amino Alcohols derived from Amino Acids

  Lüdtke, Maria Eduarda Contreira (PG)* e Diogo Seibert

  PDF - p-248-248

• Abstract - Open Access

  Further studies on the desymmetrization of cyclic olefins through the Heck-Matsuda arylation

  Angnes, Ricardo Almir; Oliveira, Caio Costa; Schwalm, Cristiane Storck; Correia, Carlos Roque Duarte

  PDF - p-249-249

• Abstract - Open Access

  Evaluation of lipases from metagenomic in kinetic resolution of secondary alcohols

  Costa, Allen C. S.; Fraiz, Talita C.; Alnoch, Robson; Madalozzo, Aline D.; Oliveira, Alfredo R. M. de; Krieger, Nadia; Piovan, Leandro

  PDF - p-250-250

• Abstract - Open Access

  Total synthesis of (±)-Preussin from an α,β-unsaturated diazoketone via the Stevens rearrangement

  Rosset, Isac G.; Burtoloso, Antonio C. B.

  PDF - p-251-251

• Abstract - Open Access

  Synthesis of Piperidines from Z-α,β-Unsaturated Diazoketones

  Rosset, Isac G.; Burtoloso, Antonio C. B.

  PDF - p-252-252

• Abstract - Open Access

  Synthesis of Simple Alkyl-Seleno-Carbohydrates

  Vargas, Jaqueline P.; Lüdtke, Diogo S.

  PDF - p-253-253

• Abstract - Open Access

  Ferrite-Nb2O5 Nanocatalyst: An Efficient Magnetically Recoverable Catalyst for Biginelli Reaction

  Lima, Carolina G. S.; Silva, Sandrina I. R. M.; Leite, Edson R.; Schwab, Ricardo S.; Corrêa, Arlene G.; Paixão, Márcio W.

  PDF - p-254-254

• Abstract - Open Access

  On the Biginelli Reaction under Homogeneous Catalysis

  Alvim, Haline G. O.; Lima, Tatiani B. de; Oliveira, Heibbe C. B.; Gozzo, Fabio C.; Macedo, Julio L.; Abdelnur, Patricia V.; Silva, Wender A.; Neto, Brenno A. D.

  PDF - p-255-255

• Abstract - Open Access

  Synthesis of a fluorescent antimicrobial peptide derivative UBI 31-38 via click reaction

  Ferreira, Soraya Maria Zandim Maciel Dias; Lara, Hugo Vinícius de Andrade; Alves, Rosemeire Brondi; Resende, Jarbas Magalhães; Freitas, Rossimiriam Pereira de

  PDF - p-256-256

• Abstract - Open Access

  Synthesis and reactivity of pyrazolo-pyridone ring, an understudied heteroaromatic scaffold

  Júnior, Paulo Eliandro da Silva; Ganesan, A.; Dale, James; Emery, Flavio

  PDF - p-257-257

• Abstract - Open Access

  Palladium-Catalyzed Direct Arylation of Selenophene

  Rampon, Daniel S.; Wessjohann, Ludger A.; Schneider, Paulo H.

  PDF - p-258-258

• Abstract - Open Access

  Chemoenzymatic Enantiospecific Synthesis of a Fluorinated myo-Inositol Analogue

  Silva, Angelo Amaro T. da; Cunha, Aline G.; Manoel, Evelin A.; Freire, Denise Maria. G.; Simas, Alessandro B. C.

  PDF - p-259-259

• Abstract - Open Access

  Synthesis and anti-HSV-1 activity of novel β-carbolines containing a substituted thiazolidin-4-one ring at C-3

  Barbosa, Valéria Aquilino; Kisukuri, Camila de Menezes; Mazia, Renata Sespede; Ueda-Nakamura, Tania; Nakamura, Celso V.; Sarragiotto*, Maria Helena

  PDF - p-260-260

• Abstract - Open Access

  Synthesis of 2-aryl-1,3-benzoselenazoles from bis(2- aminophenyl) diselenides and carboxylic acids using PBu3

  Radatz, Cátia S.; Rampon, Daniel S.; Balaguez, Renata A.; Alves, Diego; Schneider, Paulo H.

  PDF - p-261-261

• Abstract - Open Access

  Detection by ESI-MS of Negative Charge-Tagged NHC

  Rodrigues, Thyago S.; Lalli, Priscila M.; Eberlin, Marcos N.; Neto, Brenno A. D.

  PDF - p-262-262

• Abstract - Open Access

  Synthesis and evaluation of phytotoxic activity of triazole derivatives of tris(hydroxymethyl)amino methane

  Euzébio, Felipe Purisco Gomes; Alves, Rosemeire Brondi; Freitas, Rossimiriam Pereira de

  PDF - p-263-263

• Abstract - Open Access

  Selective estragole to trans-anethole isomerization in ionic liquids

  Leal, Bárbara; Pazini, Alessandra; Dupont, Jairton

  PDF - p-264-264

• Abstract - Open Access

  Rational Synthesis, Photophysical and Biochemical Evaluation of Fluorescents Chalcones as Inhibitors of Cruzain from Trypanosoma cruzi

  Silva, Wender A.; Melo, Lennine R.; Oliveira, Guilherme R.; Silva, Camilla C. C.; Trossini, Gustavo H. G.

  PDF - p-265-265

• Abstract - Open Access

  New Thiazolidine-Based Organocatalysts for Enantio- and Diastereoselective Aldol Reaction

  Jacoby, Caroline Gross; Rambo, Raoní Scheibler; Silva, Tiago Lima da; Schneider*, Paulo Henrique

  PDF - p-266-266

• Abstract - Open Access

  Synthesis of (R/S)-2-hydroxy-5-methyl-hexan-3-one, sinomone issued by Araceae species: P. acutatum and T. ulei

  Filho, Everaldo F. Santos; Maia, Artur C. D.; Navarro, Daniela M. A. F.; Princival, Jefferson L.

  PDF - p-267-267

• Abstract - Open Access

  Lipase-mediated Desymmetrization of 1,3-di-O-Benzyl-myo- Inositol

  Pais, Karla C.; Manoel, Evelin A.; Freire, Denise M. G.; Simas, Alessandro B. C.

  PDF - p-268-268

• Abstract - Open Access

  Organocatalysts: Design, Synthesis and Application in Stereoselective Domino-Michael/Henry Reactions.

  Fulas, Marcia; Figueiredo, Jéssica de S.; Rodrigues, Alessandro

  PDF - p-269-269

• Abstract - Open Access

  Synthesis of fluorescent symmetric bis-imidazolium-BTD salts

  Souza, Virginia S.; Matiello, Gabriela I.; Ferreira, Patrícia C.; Ebeling, Günter; Dupont, Jairton

  PDF - p-270-270

• Abstract - Open Access

  α,β-Unsaturated Diazoketones in Aza-Michael Additions - Application in the synthesis of Barmumycin

  Dias, Rafael Mafra de P.; Burtoloso, Antonio C. B.

  PDF - p-271-271

• Abstract - Open Access

  Design and Synthesis of Diselenides Based-Ionic Liquids

  Ferreira, Natasha L.; Nascimento, Vanessa; Braga, Antonio L.

  PDF - p-272-272

• Abstract - Open Access

  Silica-Supported Prolyl Pseudo-Peptide Organocatalysts: Application in the Direct Asymmetric Michael Addition

  Scatena, Gabriel dos S.; Torre, Alexander F. De la; Cass, Quezia B.; Paixão, Márcio W.

  PDF - p-273-273

• Abstract - Open Access

  Synthesis of triterpenes and steroids derivatives as potential anti- HIV and cancer compounds.

  Kuliakita*, Maria Candeia; Victor*, Maurício Moraes; David*, Jorge Mauricio

  PDF - p-274-274

• Abstract - Open Access

  Calixarene Catalyze Cascade Povarov−Hydrogen-Transfer Reaction in Synthesis of Quinolines

  Simões, Juliana B.; Fátima, Ângelo de; Barbosa, Luiz Claudio A.; Fernandes, Sergio A.

  PDF - p-275-275

• Abstract - Open Access

  Synthesis and identification by GC-MS of 3-(pyridin-2-yl)- thiazolidinethiones

  Mimbarcas, L.F.; Campos Jr, J.C.; Bierhals, M.P.; Cunico, W.; Siqueira, G.M.

  PDF - p-276-276

• Abstract - Open Access

  Three-Component Coupling of Amines, Aldehydes and Aliphatic Halides Under Barbier-like Conditions in Water

  Estevam, Idália Helena; Lins, Suelen; Conceição, Veronica

  PDF - p-277-277

• Abstract - Open Access

  Multicomponent catalytic Mannich Reaction: a methodological study with lawsone

  Fiorot, R. G.; Allochio Filho, J. F.; Greco, S. G.; Lacerda Jr., V.; dos Santos, R. B.; de Castro, E. V. R.

  PDF - p-278-278

• Abstract - Open Access

  Synthesis of aromatics oximes and hydrazones with electrowithdrawing substituents as reactivators of Acetylcholinesterase

  Petronilho, E. C.; Pinto, A. C.; Figueroa-Villar, J. D.

  PDF - p-279-279

• Abstract - Open Access

  Preparation and preliminiar evaluation of new organometallic bases from cis-2,6-dimethylpiperidine

  Pereira, Natália de Araujo; Soldi, Rafael Augusto; Clososki, Giuliano Cesar; Pina, Evelyn Mirella Lopes

  PDF - p-280-280

• Abstract - Open Access

  Peptide and cyclopetide synthesis via Ugi and click reactions under microwave irradiation and in continuous flow system

  Salvador, Carlos Eduardo M.; Brito, José Giovanni L.; Miranda, Leandro Soter de M.; Souza, Rodrigo O. M. A.; Andrade, Carlos Kleber Z.

  PDF - p-281-281

• Abstract - Open Access

  Synthesis of new squaramide backbone peptidomimetics catalysts

  Silva, Sandrina I. R. M.; Pozzi, Lucas; Matsuo, Bianca T.; Corrêa, Arlene G.; Paixão, Marcio W.

  PDF - p-282-282

• Abstract - Open Access

  Microwave-assisted synthesis of fused tetrazoleketopiperazine compounds via Ugi reactions

  Amaral, André Felipe C.; Silva, Wender A.; Andrade, Carlos Kleber Z.

  PDF - p-283-283

• Abstract - Open Access

  Synthesis and in vitro antifungal activity of new Mannich bases derived from 2-hydroxy-1,4-naphthoquinone (Lawsone)

  Allochio Filho, J. F.; Roldi, L. L.; Fiorot, R.; Greco, S. J.; Lacerda Jr., V.; dos Santos, R. B.; de Castro, E. V. R.; Ferreira, J. M. S.; Aleixo, A. A.; Carvalho, F. S.; Carvalho, R. S.

  PDF - p-284-284

• Abstract - Open Access

  Synthesis of new biologically actived azaspiro compounds

  Martins, Lucimara J.; Altei, Wanessa F.; Schwalm, Cristiane S.; Andricopulo, Adriano D.; Coelho, Fernando

  PDF - p-285-285

• Abstract - Open Access

  A three step continuous flow synthesis of the biaryl unit of the HIV protease inhibitor Atazanavir.

  Vechia, Luciana Dalla; Reichart, Benedikt; Glasnov, Toma; Miranda, Leandro S. M.; Kappe, C. Oliver; Souza, Rodrigo O. M. A. de

  PDF - p-286-286

• Abstract - Open Access

  New one-pot and regioselective method for the synthesis of 3-trifluoromethyl-1H-1-phenylpyrazoles

  Pittaluga, Everton P.; (PQ)*, Helio G. Bonacorso; Correa, Michele S.; Porte, Liliane M. F.; Junges, Andrizia F.; Martins, Marcos A. P.; Zanatta, Nilo

  PDF - p-287-287

• Abstract - Open Access

  SYNTHESIS OF 2,3-UNSATURATED O-GLYCOSIDES MEDIATED BY ULTRASOUND IRRADIATION

  Silva, Anderson J. Firmino Santos; Regueira, Juliana L. L. F.; Freitas, Jucleiton José R. de; Freitas, Juliano C. Rufino de; Filho, João R. de Freitas

  PDF - p-288-288

• Abstract - Open Access

  Synthesis of tetrahydropiridines by one-pot multicomponent reaction using Niobium Pentaethoxide.

  Martins, L. M.; da Silva, B. H. S. T.; Silva-Filho, L. C.

  PDF - p-289-289

• Abstract - Open Access

  Directed Metalation of Aromatic Aldimines Using Li/Mg-TMP Amides

  Cavalcante Silva, S.; Batista; H., J.; F., Moraes; Pereira; A., N. de; Clososki; G.C.

  PDF - p-290-290

• Abstract - Open Access

  New approach of side chain N-acylation and C-oxidation reactions of CF3-containing 7-amino-8-methylquinolines

  Andrighetto, Rosália; Bonacorso, Helio G.; Wiethan, Carson W.; Stefanello, Felipe S.; Martins, Marcos A. P.; Zanatta, Nilo

  PDF - p-291-291

• Abstract - Open Access

  Hydrochalcogenation of Terminal Alkynols Mediated by Zinc Organyl Chalcogenolate

  Andrade, Floyd Custódio Diniz; Matos, Gabriela Ferreira; Barros, Olga Soares do Rêgo

  PDF - p-292-292

• Abstract - Open Access

  Synthesis of 1-H-1,2,3-triazole-1,4-naphthoquinones as potential antifungal agents

  Melo, Valentina N. e; Valença, Wagner O.; Nascimento, Wilson S. do; Cordeiro, Rossana A.; Marques, Francisca J. F.; Sidrim, José Júlio C.; Camara, Celso A.; Oliveira, Ronaldo N. de

  PDF - p-293-293

• Abstract - Open Access

  Microwaves promoted an efficient synthesis of 1-thiocarbamoyl-3,5-diaryl-4,5-dihydropyrazoles

  Ritter, Marina; Rosa, Silvana Alves; Silva, Caroline Carapina da; Flores, Alex C. F.; Pizzuti, Lucas; Pereira, Claudio Martin Pereira de

  PDF - p-294-294

• Abstract - Open Access

  On the Ugi mechanism probed by ESI-MS(/MS)

  Medeiros, Gisele A.; Silva, Wender A. da; Bataglion, Giovana A.; Ferreira, Davi A. C.; Oliveira, Heibbe C. B. de; Eberlin, Marcos N.; Neto, and Brenno A. D.

  PDF - p-295-295

• Abstract - Open Access

  Synthesis of analogs of Clauraila A

  Fumagalli, Fernando; Emery, and Flavio da Silva

  PDF - p-296-296

• Abstract - Open Access

  Synthesis of 1,2,4-Triazolo[1,5-a]pyrimidine Supported under Ultrasound Irradiation

  Scapin, Elisandra; Buriol, Lilian; München, Taiana Scalco; Frizzo, Clarissa Piccinin; Martins, Marcos A. P.

  PDF - p-297-297

• Abstract - Open Access

  New phthalocyanine and azaphthalocyanine derivatives

  Svec, Jan; Zimcik, Petr

  PDF - p-298-298

• Abstract - Open Access

  Palladium complexes of aromatic bis-imines and bis-amines: synthesis and evaluation in Heck reactions.

  Andrade, Aretha P.S.; Arantes, Lucas M.; Kadooka, Juliana Y.; Carvalho, Renato L.; Fátima, Ângelo de; Sabino, Adão A.

  PDF - p-299-299

• Abstract - Open Access

  Synthesis and characterization of hydrogels from cellulose acetate by esterification crosslinking with EDTA dianhydride.

  Senna, André M.; Novak, Katia M.; Carmo, Janaina B. do; Botaro, Vagner R.

  PDF - p-300-300

• Abstract - Open Access

  Preparation of 5-Deoxypterocarpens by a-Arylation of Tetralones with o-Bromo-methoxyarenes Followed by BBr3 Mediated Cyclization

  Fernandes, Talita de A.; Domingos, Jorge L. O.; Rocha, Luiza I. A. da; Medeiros, Sabrina de; Nájera, Carmen; Costa, Paulo R. R.

  PDF - p-301-301

• Abstract - Open Access

  Chemoenzymatic resolution of fluorinated compounds by lipase CALB under microwave irradiation

  Ribeiro, Sandra S.; Guimarães, Tamara F.; Porto, André L. M.

  PDF - p-302-302

• Abstract - Open Access

  Organoselenium functionalized nitrogen heterocycles: a proposition for new antimalarials.

  Silva, Gabriela D. da; Bagnaresi, Piero; Cunha, Rodrigo L. O. R.

  PDF - p-303-303

• Abstract - Open Access

  Substrate-controlled Asymmetric Morita-Baylis-Hillman Reaction: an Approach to the Synthesis of Pyrrolizidinones and Pyrrolizidines

  Scaramal, João P. S.; Luna-Freire, Kristerson R.; Coelho, and Fernando

  PDF - p-304-304

• Abstract - Open Access

  Addition of Amino Acids to oxopyrrolidin compounds

  Ali, Bakhat; Stefani, Hélio A.; Ferreira, Fernando P.

  PDF - p-305-305

• Abstract - Open Access

  Synthesis of selenium-triazole-carbonitriles by organocatalytic cycloaddition of azidophenyl arylselenides with benzoyl nitriles.

  Seus, Natália; Sacramento, Manoela do; Savegnago, Lucielli; Alves, Diego

  PDF - p-306-306

• Abstract - Open Access

  Synthesis of Aza-Pterocarpan Analogues via 1,3 Intramolecular Dipolar Cycloadditions in in situ generated Iminoolefins

  C.F.Barcellos, Julio; Dias, Ayres G.; Sansano, José M.; Nájera, Carmen; Costa, Paulo R. R.

  PDF - p-307-307

• Abstract - Open Access

  Bromination of 4-bromoindanone and 5-bromoindanone

  Tutar, Ahmet; Yılmaz, Makbule; Erenler, Ramazan

  PDF - p-308-308